Research output per year
Research output per year
Search results
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2023
Cyclosulfamidate Mannose-Configured Cyclitol Allows Specific Allele-Dependent Inhibition of GH47 α-D-Mannosidases Through a Bump-Hole Strategy
Males, A., Kok, K., Nin-Hill, A., Beukel, S. V. D., Beenakker, T. J. M., van der Marel, G. A., Codée, J. D. C., Overkleeft, H. S., Rovira, C., Davies, G. J. & Artola, M., 17 Nov 2023, In: Chemical Science. 14, p. 13581-13586 6 p.Research output: Contribution to journal › Article › peer-review
Open AccessFile -
Human O-GlcNAcase Uses a Preactivated Boat-like Substrate Conformation for Catalysis: Evidence from X-ray Crystallography and QM/MM Metadynamics
Calvelo, M., Males, A., Alteen, M. G., Willems, L. I., Vocadlo, D. J., Davies, G. J. & Rovira, C., 10 Oct 2023, (E-pub ahead of print) In: ACS Catalysis. 13, p. 13672–13678Research output: Contribution to journal › Article › peer-review
Open AccessFile -
Structure, function and mechanism of N-glycan processing enzymes: endo-α-1,2-mannanase and endo-α-1,2-mannosidase
Burchill, L., Males, A., Kaur, A., Davies, G. J. & Williams, S. J., 1 Feb 2023, In: Israel Journal of Chemistry. 63, 1-2, 13 p., e202200067.Research output: Contribution to journal › Article › peer-review
Open AccessFile -
2022
Bicyclic picomolar OGA inhibitors enable chemoproteomic mapping of its endogenous post-translational modifications
González-Cuest, M., Sidhu, P., Ashmus, R. A., Males, A., Proceviat, C., Madden, Z., Rogalski, J. C., Busmann, J. A., Foster, L. J., Fernández, J. M. G., Davies, G. J., Mellet, C. O. & Vocadlo, D. J., 19 Jan 2022, In: Journal of the American Chemical Society. 144 , 2, p. 832–844 13 p.Research output: Contribution to journal › Article › peer-review
Open AccessFile -
2021
The development of non-hydrolysable oligosaccharide activity-based inactivators for endoglycanases: a case study on a-1,6 mannanases
Schröder, S. P., Offen, W. A., Males, A., Jin, Y., Boer, C. D., Enotarpi, J., Marino, L., van der Marel, G. A., Florea, B. I., Codée, J. D. C., Overkleeft, H. S. & Davies, G. J., 21 May 2021, (E-pub ahead of print) In: Chemistry A European Journal. 6 p.Research output: Contribution to journal › Article › peer-review
Open AccessFile