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A copper(II)-mediated radical cross-dehydrogenative coupling/sulfinic acid elimination approach to 2-quinolones
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Taylor_Quinolones_HOFQ_revised_7_10_TH_revised
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Publication details
| Journal | Tetrahedron |
|---|---|
| Date | Accepted/In press - 16 Oct 2019 |
| Date | E-pub ahead of print (current) - 21 Oct 2019 |
| Issue number | 49 |
| Volume | 75 |
| Early online date | 21/10/19 |
| Original language | English |
Abstract
A new cyclisation procedure to prepare 4-carboxy-quinolin-2-ones via a one-pot Cu(II)-mediated radical cross-dehydrogenative coupling/sulfinic acid elimination of linear anilides is described. Extensions to more complex substrates are also reported as are applications in target synthesis allowing access to natural products isolated from Oryza sativa and HOFQ.
Bibliographical note
© 2019 Elsevier Ltd. All rights reserved. This is an author-produced version of the published paper. Uploaded in accordance with the publisher’s self-archiving policy.
- 2-Quinolones, Cross-dehydrogenative coupling, Cu(II)-catalysis, Total synthesis
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