ALKYNE-ACETAL CYCLISATION REACTIONS MEDIATED BY FORMIC ACID; 3-ACYLATED-2,5-DIHYDROFURANS AND RELATED OXYGEN AND NITROGEN HETEROCYCLES

TY - JOUR

T1 - ALKYNE-ACETAL CYCLISATION REACTIONS MEDIATED BY FORMIC ACID; 3-ACYLATED-2,5-DIHYDROFURANS AND RELATED OXYGEN AND NITROGEN HETEROCYCLES

AU - Cuthbertson, James D.

AU - Godfrey, Andrew A.

AU - Unsworth, William P.

AU - Taylor, Richard J. K.

PY - 2012/1/1

Y1 - 2012/1/1

N2 - The utility of formic acid for the cyclisation of alkyne omega-acetals is described; the scope and limitations of this process are outlined and a range of acylated heterocyclic building blocks (2,5-dihydrofurans, 2,5-dihydro-1H-pyrroles, tetrahydropyridines, 2H-chromenes, 1,2-dihydroquinolines and benzoxepin5-(2H)-ones) are reported.

AB - The utility of formic acid for the cyclisation of alkyne omega-acetals is described; the scope and limitations of this process are outlined and a range of acylated heterocyclic building blocks (2,5-dihydrofurans, 2,5-dihydro-1H-pyrroles, tetrahydropyridines, 2H-chromenes, 1,2-dihydroquinolines and benzoxepin5-(2H)-ones) are reported.

UR - http://www.scopus.com/inward/record.url?scp=84856515341&partnerID=8YFLogxK

U2 - 10.3987/COM-11-S(P)79

DO - 10.3987/COM-11-S(P)79

M3 - Article

SN - 0385-5414

VL - 84

SP - 1013

EP - 1021

JO - Heterocycles

JF - Heterocycles

IS - 2

ER -