Preparation of 2-substituted benzimidazoles and related heterocycles directly from activated alcohols using TOP methodology

C D  Wilfred; R J K  Taylor

doi:10.1055/s-2004-829060

Preparation of 2-substituted benzimidazoles and related heterocycles directly from activated alcohols using TOP methodology

C D Wilfred, R J K Taylor

Chemistry

Research output: Contribution to journal › Article › peer-review

Abstract

A one-pot procedure for preparing 2-substituted benzimidazoles directly from activated alcohols in good to excellent yields using a new Tandem Oxidation Process (TOP) is reported. The use of this methodology to prepare 2-substituted benzoxazoles and 2-substituted benzothiazoles is also described.

Original language	English
Pages (from-to)	1628-1630
Number of pages	3
Journal	Synlett
Issue number	9
DOIs	https://doi.org/10.1055/s-2004-829060
Publication status	Published - 22 Jul 2004

Keywords

2-substituted benzimidazoles
2-substituted benzoxazoles
2-substituted benzothiazoles
Tandem Oxidation Procedure
one-pot

Access to Document

10.1055/s-2004-829060

Cite this

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title = "Preparation of 2-substituted benzimidazoles and related heterocycles directly from activated alcohols using TOP methodology",

abstract = "A one-pot procedure for preparing 2-substituted benzimidazoles directly from activated alcohols in good to excellent yields using a new Tandem Oxidation Process (TOP) is reported. The use of this methodology to prepare 2-substituted benzoxazoles and 2-substituted benzothiazoles is also described.",

keywords = "2-substituted benzimidazoles, 2-substituted benzoxazoles, 2-substituted benzothiazoles, Tandem Oxidation Procedure, one-pot",

author = "Wilfred, {C D} and Taylor, {R J K}",

year = "2004",

month = jul,

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doi = "10.1055/s-2004-829060",

language = "English",

pages = "1628--1630",

journal = "Synlett",

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publisher = "Georg Thieme Verlag",

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AU - Wilfred, C D

AU - Taylor, R J K

PY - 2004/7/22

Y1 - 2004/7/22

N2 - A one-pot procedure for preparing 2-substituted benzimidazoles directly from activated alcohols in good to excellent yields using a new Tandem Oxidation Process (TOP) is reported. The use of this methodology to prepare 2-substituted benzoxazoles and 2-substituted benzothiazoles is also described.

AB - A one-pot procedure for preparing 2-substituted benzimidazoles directly from activated alcohols in good to excellent yields using a new Tandem Oxidation Process (TOP) is reported. The use of this methodology to prepare 2-substituted benzoxazoles and 2-substituted benzothiazoles is also described.

KW - 2-substituted benzimidazoles

KW - 2-substituted benzoxazoles

KW - 2-substituted benzothiazoles

KW - Tandem Oxidation Procedure

KW - one-pot

U2 - 10.1055/s-2004-829060

DO - 10.1055/s-2004-829060

M3 - Article

SN - 1437-2096

SP - 1628

EP - 1630

JO - Synlett

JF - Synlett

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