THE PREPARATION OF NOVEL DOPAMINE ANALOGS VIA PALLADIUM CATALYZED CYCLIZATION REACTIONS

A J  DAVIES; R J K  TAYLOR; D I  SCOPES; A H  WADSWORTH

doi:10.1016/S0960-894X(00)80174-2

THE PREPARATION OF NOVEL DOPAMINE ANALOGS VIA PALLADIUM CATALYZED CYCLIZATION REACTIONS

A J DAVIES, R J K TAYLOR, D I SCOPES, A H WADSWORTH

Chemistry

Research output: Contribution to journal › Article › peer-review

Abstract

The preparation of a range of tetrahydronaphthalene derivatives via palladium catalysed cyclisation reactions is described. The application of the cyclisation methodology to the synthesis of enantiomerically pure amino-chromans, as potential dopamine analogues, is also discussed.

Original language	English
Pages (from-to)	481-484
Number of pages	4
Journal	Bioorganic & Medicinal Chemistry Letters
Volume	2
Issue number	5
DOIs	https://doi.org/10.1016/S0960-894X(00)80174-2
Publication status	Published - May 1992

Keywords

ANION CAPTURE PROCESSES
PHARMACOLOGY
DERIVATIVES

Access to Document

10.1016/S0960-894X(00)80174-2

Cite this

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title = "THE PREPARATION OF NOVEL DOPAMINE ANALOGS VIA PALLADIUM CATALYZED CYCLIZATION REACTIONS",

abstract = "The preparation of a range of tetrahydronaphthalene derivatives via palladium catalysed cyclisation reactions is described. The application of the cyclisation methodology to the synthesis of enantiomerically pure amino-chromans, as potential dopamine analogues, is also discussed.",

keywords = "ANION CAPTURE PROCESSES, PHARMACOLOGY, DERIVATIVES",

author = "DAVIES, {A J} and TAYLOR, {R J K} and SCOPES, {D I} and WADSWORTH, {A H}",

year = "1992",

month = may,

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journal = "Bioorganic & Medicinal Chemistry Letters",

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AU - DAVIES, A J

AU - TAYLOR, R J K

AU - SCOPES, D I

AU - WADSWORTH, A H

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N2 - The preparation of a range of tetrahydronaphthalene derivatives via palladium catalysed cyclisation reactions is described. The application of the cyclisation methodology to the synthesis of enantiomerically pure amino-chromans, as potential dopamine analogues, is also discussed.

AB - The preparation of a range of tetrahydronaphthalene derivatives via palladium catalysed cyclisation reactions is described. The application of the cyclisation methodology to the synthesis of enantiomerically pure amino-chromans, as potential dopamine analogues, is also discussed.

KW - ANION CAPTURE PROCESSES

KW - PHARMACOLOGY

KW - DERIVATIVES

U2 - 10.1016/S0960-894X(00)80174-2

DO - 10.1016/S0960-894X(00)80174-2

M3 - Article

SN - 0960-894X

VL - 2

SP - 481

EP - 484

JO - Bioorganic & Medicinal Chemistry Letters

JF - Bioorganic & Medicinal Chemistry Letters

IS - 5

ER -